Fig. 8.
Effects of the intravenous administration of DOI on serotonergic neurons of the DR. A–E, Integrated firing rate histograms showing the effect of DOI on five different 5-HT neurons. A–C depict neurons with full (A) and partial (B, C) inhibitory responses to the administration of cumulative doses of DOI (25–50 μg/kg, i.v. in A; 25–400 μg/kg, i.v. inB, C). The effect of DOI was antagonized by M100907 (100 μg/kg, i.v.; examples in B andD). The serotonergic nature of neurons with partial or full response to DOI is illustrated by its sensitivity to 8-OH-DPAT (C, D). D shows the inhibitory effect of DOI (25–50 μg/kg, i.v.). After reversal by M100907 (100 μg/kg, i.v.), 8-OH-DPAT (DPAT; 0.25–2 μg/kg, i.v.) fully suppressed firing activity, and the 5-HT1A receptor antagonist WAY 100635 (WAY; 10 μg/kg, i.v.) returned firing rate to baseline. E shows the reversal of the effect of DOI (25–200 μg/kg, i.v.) by the GABAAantagonist picrotoxinin (PTX; 1 mg/kg, i.v.). The graph inF shows the dose–response curves for DOI in 5-HT neurons. The neurons with partial and full inhibitory responses to DOI administration had comparable ED50 values (19 and 22 μg/kg, i.v.; n = 7 and 5, respectively). Thedotted line shows the dose–response curve for all neurons (n = 12).