Table 2. Binding ability of ligands to mutant and wild-type CbuqPBP1.
Ligands | IC50 (µM) | Ki (µM) | ||||
---|---|---|---|---|---|---|
PBP1 | H53A | F69A | PBP1 | H53A | F69A | |
benzothiazole | 13.426 | – | 10.538 | 9.822 | – | 7.305 |
dibutyl phthalate | 16.889 | – | 20.04 | 12.355 | – | 13.893 |
cedrol | 29.953 | – | – | 21.912 | – | – |