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. 2019 Oct 17;9:14907. doi: 10.1038/s41598-019-51445-w

Table 2.

Tumor-to-organ ratios of in BALB/C nu/nu mice bearing SK-RC-52 OV xenografts.

[111In]In-DOTA-HE3-ZCAIX:2 [99mTc]Tc(CO)3-HE3-ZCAIX:2 [111In]In-DTPA-G250(Fab’)2 [111In]In-DTPA-G250(Fab’)2
4 h 4 h 4 h 24 h
Blood 63 ± 11a 23 ± 2d,e 2.1 ± 0.2b 67 ± 12
Lung 30 ± 3a 16 ± 2d,e 2.7 ± 0.4b 7 ± 1c
Liver 33 ± 2a 8 ± 2d,e 0.7 ± 0.3b 0.6 ± 0.2c
Spleen 37 ± 3a 24 ± 6d,e 0.7 ± 0.2b 0.6 ± 0.2c
Stomach 36 ± 4a 22 ± 6d,e 4.4 ± 0.6b 6 ± 3c
Duodenum 31 ± 8 19 ± 6d,e 2.4 ± 1.2b 3 ± 2c
Kidney 0.038 ± 0.008 0.04 ± 0.01d 0.029 ± 0.005 0.03 ± 0.01
Muscle 102 ± 20a 62 ± 6d,e 7.9 ± 0.7b 11 ± 1c
Bone 47 ± 8a 28 ± 3d,e 3.0 ± 0.5b 4 ± 1c

Results are presented as %ID/g (the mean values and standard deviation for four mice).

aSignificant difference (p < 0.05) between [111In]In-DOTA-ZCAIX:2 and [99mTc]Tc(CO)3-HE3-ZCAIX:2;

bSignificant difference (p < 0.05) between [111In]In-DOTA-ZCAIX:2 and [111In]In-G250(Fab’)2 (4 h);

cSignificant difference (p < 0.05) between [111In]In-DOTA-ZCAIX:2 and [111In]In-G250(Fab’)2 (24 h);

dSignificant difference (p < 0.05) between [99mTc]Tc(CO)3-HE3-ZCAIX:2 and [111In]In-G250(Fab’)2 (4 h);

eSignificant difference (p < 0.05) between [99mTc]Tc(CO)3-HE3-ZCAIX:2 and [111In]In-G250(Fab’)2 (4 h).