Table 2. Comparison of apparent activation constants (Kact) for four PKA isoforms obtained by in vitro biochemical kinase assay.
Kact [µM] | ||||
---|---|---|---|---|
PKA-Iα | PKA-Iβ | PKA-IIα | PKA-IIβ | |
cAMP | 0.085 | 0.038 | 0.080 | 0.19 |
007 | 14 | 18 | >70 | 50 |
S-220 | 0.29 | 0.29 | 0.27 | 0.21 |
S-223 | >1000 | >1000 | >25 | >1000 |