Table 5.

Type III ATX inhibitors based on their kinetic and crystallographic analysis.

	Type III Inhibitor	PDB ID	Activity (IC50)	Reference
7-α-hydroxycholesterol		5dlt	undetermined	[26]
TUDCA		5dlw	10.4 µM	[26]
PAT-347		4zg7	0.3 nM	[50]
PAT-505		5kxa	2 nM	[70]
LM-Cpd 51		5lqq	81 nM	[71]