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. 2019 Oct 24;6(Pt 6):1106–1119. doi: 10.1107/S2052252519013137

Table 2. β2AR ligands used in the exchange experiments with their MoAs, molecular weights (MW) and affinity (K i) values.

Data are from the ChEMBL database (ChEMBL_23; Gaulton et al., 2012). Chemical structures of the ligands used for the other receptors in this study are shown in Supplementary Fig. S4.

Ligand Chemical structure MoA ChEMBL ID MW (Da) K i (nM) Reference
ICI-118,551 graphic file with name m-06-01106-scheme1.jpg Inverse agonist CHEMBL513389 277.4 0.13 Dolušić et al. (2011)
Carazolol graphic file with name m-06-01106-scheme2.jpg Inverse agonist CHEMBL324665 298.4 0.114 Sabio et al. (2008)
Timolol graphic file with name m-06-01106-scheme3.jpg Inverse agonist CHEMBL499 316.4 0.201  
Propranolol graphic file with name m-06-01106-scheme4.jpg Inverse agonist CHEMBL27 259.3 3.69 Plazinska et al. (2014)
Alprenolol graphic file with name m-06-01106-scheme5.jpg Antagonist CHEMBL266195 249.4 1 Aristotelous et al. (2013)
Carvedilol graphic file with name m-06-01106-scheme6.jpg β-Arrestin-biased agonist CHEMBL723 406.5 0.166  
Procaterol graphic file with name m-06-01106-scheme7.jpg Agonist CHEMBL160519 290.4 78 Baker (2010)
Formoterol graphic file with name m-06-01106-scheme8.jpg Agonist CHEMBL3989798 344.4 23 Baker (2010)

Values are from the DrugMatrix Database (https://ntp.niehs.nih.gov/drugmatrix/index.html).