Table 1.
Entry | Cyclic Nitrone | Pyrrolidine | Yield a | Alcohol | Product | Yield b |
---|---|---|---|---|---|---|
1 | 64% | 43% | ||||
2 | 43% | |||||
3 | 65% | 41% | ||||
4 | 45% | |||||
5 | 64% | 40% | ||||
6 | 41% | |||||
7 | 71% | 43% | ||||
8 | 43% |
a Total yield in 3 steps starting from cyclic nitrones to the corresponding pyrrolidine. b Total yield in 2 steps starting from pyrrolidine cores to broussonetine M or its analogues.