Table 3. Biodistribution (% ID per g) of the Bi3+ complexes with H4DOTA and H4BATA in normal mice a .
| Tissue | [207Bi]DOTA-Bi |
[207Bi]BATA-Bi |
||
| Time points (h) | ||||
| 1 | 6 | 1 | 6 | |
| Kidneys | 1.83 ± 0.42 | 1.10 ± 0.23 | 3.03 ± 0.52 | 1.97 ± 0.14 |
| Blood | 1.22 ± 0.29 | b | 1.14 ± 0.63 | b |
| Femur | 0.97 ± 0.60 | 0.14 ± 0.07 | 0.58 ± 0.23 | 0.07 ± 0.01 |
| Liver | 0.18 ± 0.02 | 0.07 ± 0.01 | 0.40 ± 0.29 | 0.11 ± 0.02 |
| Heart | 0.07 ± 0.01 | b | 0.10 ± 0.08 | 0.02 ± 0.01 |
| Lungs | 0.16 ± 0.03 | 0.03 ± 0.01 | 0.22 ± 0.13 | 0.06 ± 0.01 |
| Spleen | 0.12 ± 0.01 | 0.04 ± 0.02 | 0.19 ± 0.13 | 0.08 ± 0.02 |
| Brain | 0.05 ± 0.01 | b | 0.02 ± 0.01 | b |
| The rest of body | 0.47 ± 0.09 | 0.15 ± 0.01 | 1.1 ± 0.5 | 0.25 ± 0.06 |
a n = 3 for each point.
bRadioactivity is lower than the minimum detectable level.