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. 2019 Nov 11;176(Suppl 1):S229–S246. doi: 10.1111/bph.14750
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=605 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=606 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=607
Systematic nomenclature NR1I1 NR1I2 NR1I3
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:12679, http://www.uniprot.org/uniprot/P11473 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:7968, http://www.uniprot.org/uniprot/O75469 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:7969, http://www.uniprot.org/uniprot/Q14994
Endogenous agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2779 [http://www.ncbi.nlm.nih.gov/pubmed/7976510?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/12089348?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=1013 [http://www.ncbi.nlm.nih.gov/pubmed/10628745?dopt=AbstractPlus]
Selective agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2777 [http://www.ncbi.nlm.nih.gov/pubmed/1472092?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/8573413?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2790 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2764 [http://www.ncbi.nlm.nih.gov/pubmed/10852961?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/10974665?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2759 [http://www.ncbi.nlm.nih.gov/pubmed/10628745?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2739 [http://www.ncbi.nlm.nih.gov/pubmed/9727070?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2765 [http://www.ncbi.nlm.nih.gov/pubmed/9784494?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/9727070?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2756 [http://www.ncbi.nlm.nih.gov/pubmed/10757780?dopt=AbstractPlus] – Mouse, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2758 [http://www.ncbi.nlm.nih.gov/pubmed/12611900?dopt=AbstractPlus]
Selective antagonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2788 (pIC50 8.2) [http://www.ncbi.nlm.nih.gov/pubmed/17125259?dopt=AbstractPlus] – Chicken, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2789 (pIC50 7.5) [http://www.ncbi.nlm.nih.gov/pubmed/12901907?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/11094341?dopt=AbstractPlus]
Comments http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2330 [http://www.ncbi.nlm.nih.gov/pubmed/10748001?dopt=AbstractPlus] and http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2755 [http://www.ncbi.nlm.nih.gov/pubmed/23665929?dopt=AbstractPlus] although acting at other sites, function as antagonists of the constitutive androstane receptor.