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. 2019 Nov 11;176(Suppl 1):S247–S296. doi: 10.1111/bph.14751
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1905 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1906 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1907 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2321 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1908
Subunits http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1734 (Ligand‐binding subunit), http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1897 (Other subunit) http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1735 (Ligand‐binding subunit), http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1897 (Other subunit) http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1736 (Ligand‐binding subunit), http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1897 (Other subunit) http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2319 (Ligand‐binding subunit), http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1897 (Other subunit) http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1737 (Ligand‐binding subunit), http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2320 (Other subunit)
Inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6972 (pK d 7.8) [http://www.ncbi.nlm.nih.gov/pubmed/1834644?dopt=AbstractPlus]
Endogenous agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4973 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:5991, http://www.uniprot.org/uniprot/P01583), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4974 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:5992, http://www.uniprot.org/uniprot/P01584) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5880 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:16028, http://www.uniprot.org/uniprot/O95760) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5881 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15562, http://www.uniprot.org/uniprot/Q9UHA7), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5882 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15564, http://www.uniprot.org/uniprot/Q9NZH7), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5883 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15741, http://www.uniprot.org/uniprot/Q9NZH8) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4983 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:5986, http://www.uniprot.org/uniprot/Q14116), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6149 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15563, http://www.uniprot.org/uniprot/Q9NZH6)
Endogenous antagonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5878 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6000, http://www.uniprot.org/uniprot/P18510) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5879 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15561, http://www.uniprot.org/uniprot/Q9UBH0)
Selective antagonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4861 [http://www.ncbi.nlm.nih.gov/pubmed/8940020?dopt=AbstractPlus]
Comments http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5879 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15561, http://www.uniprot.org/uniprot/Q9UBH0) is a highly specific antagonist of the response to http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5883 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:15741, http://www.uniprot.org/uniprot/Q9NZH8). Decoy receptor that binds http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4973 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:5991, http://www.uniprot.org/uniprot/P01583), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4974 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:5992, http://www.uniprot.org/uniprot/P01584) and http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5878 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6000, http://www.uniprot.org/uniprot/P18510).