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. 2019 Nov 11;176(Suppl 1):S247–S296. doi: 10.1111/bph.14751
Nomenclature https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2450 https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2451 https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2452 https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2453 https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2454 https://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2455
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6147, http://www.uniprot.org/uniprot/P38570 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6148, http://www.uniprot.org/uniprot/P20701 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6149, http://www.uniprot.org/uniprot/P11215 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6150, http://www.uniprot.org/uniprot/P06756 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6152, http://www.uniprot.org/uniprot/P20702 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6153, http://www.uniprot.org/uniprot/P05556
Antagonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=7533 (Inhibition) [18, http://www.ncbi.nlm.nih.gov/pubmed/24900456?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=9689 (pIC50 7.1) [http://www.ncbi.nlm.nih.gov/pubmed/14561098?dopt=AbstractPlus]
Antibodies http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6593 (Binding) (pK d 11.4) [100]