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. 2019 Nov 11;176(Suppl 1):S247–S296. doi: 10.1111/bph.14751
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1850 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1851 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1852 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1853 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1854 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1855 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1856
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9664, http://www.uniprot.org/uniprot/P18433 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9665, http://www.uniprot.org/uniprot/P23467 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9666, http://www.uniprot.org/uniprot/P08575 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9668, http://www.uniprot.org/uniprot/P23468 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9669, http://www.uniprot.org/uniprot/P23469 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9670, http://www.uniprot.org/uniprot/P10586 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9671, http://www.uniprot.org/uniprot/P23470
Putative endogenous ligands http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6603 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6561, http://www.uniprot.org/uniprot/P09382) [http://www.ncbi.nlm.nih.gov/pubmed/10369126?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6607 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:25042, http://www.uniprot.org/uniprot/Q9NT99) [http://www.ncbi.nlm.nih.gov/pubmed/20139422?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6607 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:25042, http://www.uniprot.org/uniprot/Q9NT99) [http://www.ncbi.nlm.nih.gov/pubmed/20139422?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6609 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:2173, http://www.uniprot.org/uniprot/Q9P232), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6612 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:2174, http://www.uniprot.org/uniprot/Q8IWV2), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6613 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:2175, http://www.uniprot.org/uniprot/O94779), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6614 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:2176, http://www.uniprot.org/uniprot/Q9UQ52) [http://www.ncbi.nlm.nih.gov/pubmed/20133774?dopt=AbstractPlus]
Inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=8770 (pIC50 5.9) [http://www.ncbi.nlm.nih.gov/pubmed/18579388?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=8831 (pK i 5.6) [http://www.ncbi.nlm.nih.gov/pubmed/21882820?dopt=AbstractPlus]