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. 2019 Nov 11;176(Suppl 1):S247–S296. doi: 10.1111/bph.14751
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1876 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1877 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1878 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1879 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1880 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2323 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2324
Systematic nomenclature TNFRSF7 TNFRSF8 TNFRSF9 TNFRSF10A TNFRSF10B TNFRSF10C TNFRSF10D
Common abbreviation DR4 DR5
HGNC, UniProt http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1876, http://www.uniprot.org/uniprot/P26842 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11923, http://www.uniprot.org/uniprot/P28908 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11924, http://www.uniprot.org/uniprot/Q07011 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11904, http://www.uniprot.org/uniprot/O00220 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11905, http://www.uniprot.org/uniprot/O14763 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11906, http://www.uniprot.org/uniprot/O14798 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11907, http://www.uniprot.org/uniprot/Q9UBN6
Adaptor proteins TRAF2, SIVA TRAF1, TRAF2, TRAF3, TRAF5 TRAF1, TRAF2, TRAF3 FADD FADD
Endogenous ligands https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11937 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11937, http://www.uniprot.org/uniprot/P32970) http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1877 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11938, http://www.uniprot.org/uniprot/P32971) http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1878 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11939, http://www.uniprot.org/uniprot/P41273) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5065 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11925, http://www.uniprot.org/uniprot/P50591)
Endogenous agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5065 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11925, http://www.uniprot.org/uniprot/P50591) [251]
Agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=8889 [81]
Antibodies http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6772 (Inhibition) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=9334 (Agonist) (pK d ~8.5) [251]
Comments Decoy receptor for http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5065 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11925, http://www.uniprot.org/uniprot/P50591). Decoy receptor for http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5065 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:11925, http://www.uniprot.org/uniprot/P50591).