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. 2019 Nov 11;176(Suppl 1):S297–S396. doi: 10.1111/bph.14752
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2358 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2394 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2392 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2397 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2424
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:3309, http://www.uniprot.org/uniprot/P08246 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9071, http://www.uniprot.org/uniprot/P00747 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9051, http://www.uniprot.org/uniprot/P00750 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:9475, http://www.uniprot.org/uniprot/P07477 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:12019, http://www.uniprot.org/uniprot/Q15661
EC number http://www.genome.jp/dbget‐bin/www_bget?ec:3.4.21.37 http://www.genome.jp/dbget‐bin/www_bget?ec:3.4.21.7 http://www.genome.jp/dbget‐bin/www_bget?ec:3.4.21.68 http://www.genome.jp/dbget‐bin/www_bget?ec:3.4.21.4 http://www.genome.jp/dbget‐bin/www_bget?ec:3.4.21.59
Inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6476 (pK i 8) [http://www.ncbi.nlm.nih.gov/pubmed/21791628?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6441 (pIC50 7.4) [http://www.ncbi.nlm.nih.gov/pubmed/21741848?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6570 {Bovine} (Binding) (pIC50 6.8) [http://www.ncbi.nlm.nih.gov/pubmed/17666018?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6573 (Binding) (pIC50 3.6) [http://www.ncbi.nlm.nih.gov/pubmed/17666018?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4262 (pIC50 7.8) [http://www.ncbi.nlm.nih.gov/pubmed/9544206?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4262 (pIC50 10) [http://www.ncbi.nlm.nih.gov/pubmed/12939527?dopt=AbstractPlus]
Selective inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=6574 (Binding) (pIC50 4.4) [http://www.ncbi.nlm.nih.gov/pubmed/24900876?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=7863 (pIC50 8.5) [http://www.ncbi.nlm.nih.gov/pubmed/11172730?dopt=AbstractPlus]