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. 2019 Nov 11;176(Suppl 1):S297–S396. doi: 10.1111/bph.14752
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1294 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1295 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1296
Common abbreviation PDE1A PDE1B PDE1C
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:8774, http://www.uniprot.org/uniprot/P54750 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:8775, http://www.uniprot.org/uniprot/Q01064 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:8776, http://www.uniprot.org/uniprot/Q14123
EC number http://www.genome.jp/dbget‐bin/www_bget?ec:3.1.4.17 http://www.genome.jp/dbget‐bin/www_bget?ec:3.1.4.17 http://www.genome.jp/dbget‐bin/www_bget?ec:3.1.4.17
Rank order of affinity http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2347 > http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2352 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2347 > http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2352 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2347 = http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2352
Endogenous activators http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2351 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1442 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1445 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1449, http://www.uniprot.org/uniprot/P62158) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2351 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1442 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1445 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1449, http://www.uniprot.org/uniprot/P62158) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2351 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1442 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1445 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:1449, http://www.uniprot.org/uniprot/P62158)
Endogenous inhibitors
Inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=9151 (pIC50 5.2) [http://www.ncbi.nlm.nih.gov/pubmed/19303290?dopt=AbstractPlus]
Sub/family‐selective inhibitors
Selective inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5270 (pIC50 7.2) [http://www.ncbi.nlm.nih.gov/pubmed/8961086?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5285 (pIC50 5.1) [http://www.ncbi.nlm.nih.gov/pubmed/8557689?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5270 (pIC50 7.2) [http://www.ncbi.nlm.nih.gov/pubmed/8961086?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5270 (pIC50 7.2) [http://www.ncbi.nlm.nih.gov/pubmed/8961086?dopt=AbstractPlus], vinpocetine (pIC50 4.3) [http://www.ncbi.nlm.nih.gov/pubmed/8557689?dopt=AbstractPlus]
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