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. 2019 Nov 11;176(Suppl 1):S297–S396. doi: 10.1111/bph.14752
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1433 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1434
HGNC, UniProt http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1433, http://www.uniprot.org/uniprot/Q13393 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=1434, http://www.uniprot.org/uniprot/O14939
EC number http://www.genome.jp/dbget‐bin/www_bget?ec:3.1.4.4 http://www.genome.jp/dbget‐bin/www_bget?ec:3.1.4.4 A phosphatidylcholine + H2O <=> choline + a phosphatidate
Endogenous activators http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5305 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:652, http://www.uniprot.org/uniprot/P84077), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2387, RhoA, PKC evoked phosphorylation, RalA [http://www.ncbi.nlm.nih.gov/pubmed/9013646?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/9207251?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5305 (https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:652, http://www.uniprot.org/uniprot/P84077), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2387 [http://www.ncbi.nlm.nih.gov/pubmed/9582313?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=1054 [http://www.ncbi.nlm.nih.gov/pubmed/12374567?dopt=AbstractPlus]
Endogenous inhibitors Gßγ [http://www.ncbi.nlm.nih.gov/pubmed/16638972?dopt=AbstractPlus] Gßγ [http://www.ncbi.nlm.nih.gov/pubmed/16638972?dopt=AbstractPlus]
Inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=8781 (pIC50 8) [http://www.ncbi.nlm.nih.gov/pubmed/19136975?dopt=AbstractPlus] –
Selective inhibitors http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=8782 (pIC50 7.3) [http://www.ncbi.nlm.nih.gov/pubmed/19136975?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=5287 (pIC50 7.7) [http://www.ncbi.nlm.nih.gov/pubmed/20735042?dopt=AbstractPlus]