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. 2019 Nov 11;176(Suppl 1):S142–S228. doi: 10.1111/bph.14749
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=416 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=417 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=418 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=419
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:4084, http://www.uniprot.org/uniprot/O14764 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:4085, http://www.uniprot.org/uniprot/P78334 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:14454, http://www.uniprot.org/uniprot/Q9UN88 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:4089, http://www.uniprot.org/uniprot/O00591
Selective agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4322 [GABA site]
Channel blockers http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051
Comments http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=566 is an endogenous allosteric regulator and causes potent inhibition of receptors formed from binary combinations of α and β subunits, incorporation of a δ or γ subunit causes a modest, or pronounced, reduction in inhibitory potency, respectively