Skip to main content
. 2019 Nov 11;176(Suppl 1):S142–S228. doi: 10.1111/bph.14749
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=420 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=421 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=422
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:4090, http://www.uniprot.org/uniprot/P24046 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:4091, http://www.uniprot.org/uniprot/P28476 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:17969, http://www.uniprot.org/uniprot/A8MPY1
Agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4226 [GABA site] (Partial agonist), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4259 [GABA site] (Partial agonist) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4226 [GABA site] (Partial agonist), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4259 [GABA site] (Partial agonist) http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4226 [GABA site] (Partial agonist), http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4259 [GABA site] (Partial agonist)
Selective agonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4067 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4107 [GABA site] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4067 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4107 [GABA site] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4067 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4107 [GABA site]
Antagonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4322 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4227 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4287 [GABA site] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4322 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4227 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4287 [GABA site] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4322 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4227 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4287 [GABA site]
Selective antagonists http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4096 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4099 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4328 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4143 [GABA site] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4096 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4099 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4328 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4143 [GABA site] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4096 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4099 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4328 [GABA site], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4143 [GABA site]
Channel blockers http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051 http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4320, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=4051
Comments http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2312 is not active at this subunit http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2312 is not active at this subunit http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2312 is not active at this subunit