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. 2019 Nov 11;176(Suppl 1):S142–S228. doi: 10.1111/bph.14749
Nomenclature http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=545 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=546 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=547 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=548 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=549 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=550 http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=551
HGNC, UniProt https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6219, http://www.uniprot.org/uniprot/Q16322 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6231, http://www.uniprot.org/uniprot/Q14721 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6232, http://www.uniprot.org/uniprot/Q92953 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6233, http://www.uniprot.org/uniprot/P48547 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6234, http://www.uniprot.org/uniprot/Q96PR1 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6235, http://www.uniprot.org/uniprot/Q14003 https://www.genenames.org/data/gene‐symbol‐report/#!/hgnc_id/HGNC:6236, http://www.uniprot.org/uniprot/Q03721
Associated subunits Kv β1 and Kv β2 Kv5.1, Kv6.1‐6.4, Kv8.1‐8.2 and Kv9.1‐9.3 Kv5.1, Kv6.1‐6.4, Kv8.1‐8.2 and Kv9.1‐9.3 MiRP2 is an associated subunit for Kv3.4
Channel blockers http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2416 (pIC50 2.8) [http://www.ncbi.nlm.nih.gov/pubmed/10836990?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2343 (Pore blocker) (pIC50 2) [http://www.ncbi.nlm.nih.gov/pubmed/16478442?dopt=AbstractPlus] – Rat http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2416 (pIC50 2.8) [http://www.ncbi.nlm.nih.gov/pubmed/9612272?dopt=AbstractPlus], http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2343 (pIC50 2.6) [http://www.ncbi.nlm.nih.gov/pubmed/9612272?dopt=AbstractPlus] http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2416 (pIC50 4.5) [http://www.ncbi.nlm.nih.gov/pubmed/7517498?dopt=AbstractPlus] – Mouse, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2343 (pIC50 3.7) [http://www.ncbi.nlm.nih.gov/pubmed/7517498?dopt=AbstractPlus] – Mouse http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2416 (pIC50 4.6) [http://www.ncbi.nlm.nih.gov/pubmed/11790809?dopt=AbstractPlus] – Rat, http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2343 (pIC50 4.2) [http://www.ncbi.nlm.nih.gov/pubmed/11790809?dopt=AbstractPlus] – Rat http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2343 (pIC50 3.9) [http://www.ncbi.nlm.nih.gov/pubmed/1381835?dopt=AbstractPlus] – Rat http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2343 (pIC50 3.5) [http://www.ncbi.nlm.nih.gov/pubmed/1378392?dopt=AbstractPlus, http://www.ncbi.nlm.nih.gov/pubmed/1840526?dopt=AbstractPlus] – Rat
Selective channel blockers http://www.guidetopharmacology.org/GRAC/LigandDisplayForward?ligandId=2578 (pIC50 7.3) [http://www.ncbi.nlm.nih.gov/pubmed/9506974?dopt=AbstractPlus] – Rat
Functional Characteristics KV KV KV KV KA KA