Table 1. Correlation of docking simulation results with in vitro conjugation capacity of UGT1A1.
Substrate | Correct binding mode of UDPGA | Hydroxyl orientation of substrate | ||
---|---|---|---|---|
Correlation coefficient | P value | Correlation coefficient | P value | |
AAP | - 0.189 | 0.7195, >0.05 | 0.954 | 0.0032, <0.01 |
E2 | 0.114 | 0.8298, >0.05 | 0.994 | 0.00005, <0.001 |