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. Author manuscript; available in PMC: 2019 Nov 18.
Published in final edited form as: Future Drug Discov. 2019 Sep 2;1(2):FDD17. doi: 10.4155/fdd-2019-0022

Table 1.

Preliminary biological data for JT09.

Peripheral selectivity >938-fold
Kappa over mu or delta selectivity >33,400-fold
Oral ED50 4.7 mg/kg
Intravenous ED50 0.032 mg/kg