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. 2019 Oct 31;10(11):1543–1548. doi: 10.1021/acsmedchemlett.9b00377

Table 4. HBE-TECC and CYP3A4 Induction SAR for Aromatic Analogs 10 and 1217.

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a

HBE-TECC assay using ABBV-2222 (0.15 μM) and GLPG1837 (0.75 μM) as the positive controls. All values are the geometric means of at least two determinations.

b

All values are the means of at least three determinations.