Animals with tumor received 4 doses of TXT-NPs (12 mg/kg TXT
dose-equivalent NPs) in combination with DNmb (3 mg/kg), both given simultaneous
as an IV injection. The other groups were DNmb alone (3 mg/kg, as IV injection),
TXT-Cremophor (12 mg/kg), and saline (n=3). Arrows indicate dosing schedule.
Changes in a) bioluminance signal; p<0.05 (each group
compared with saline group); b) body weight, p<0.05 for both
DNmb and combination treatment when compared with saline control; TXT Cr-EL
group shows no statistical significance with saline control; c)
survival with time; and d) representative bioluminance images of
untreated, TXT-NPs and the combination (DNmb+TXT-NPs) treated animals.
Combination vs. other groups, p=0.01. Saline, vs. TXT Cr-EL or DNmb p=NS. Data
are expressed as the mean ± s.e.m., n= 3 to 5. The combination treatment
was most effective in terms of tumor regression, body weight gain, and survival
as compared with other treatment groups. There was no tumor relapse in the
combination group even after discontinuing the treatment, whereas DNmb alone
treated group showed tumor relapse. Median survival for saline = 7 wks; DNmb =14
wks; TXT-Cr-EL = 9 wks; and DNmb + TXT-NP > 40 wks, which is beyond the
study end point. Abbreviation, D is for days, whereas other time points are in
weeks.