Table 2.
MCT1 IC50 (nM) values of CHC derivatives 2a–d.
| Compound | MCT1 |
|---|---|
| CHC 1 | >150000 |
| TBDPS-CHC 2a | 408 ± 5 |
| Ex-TBDPS-CHC 2b | 97 ± 7 |
| Ex-OH-CHC 2c | >5000 |
| Ex-Br-CHC 2d | >5000 |
*Average ± SEM of three separate experiments.
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