| ABMECA | N6-(4-Aminobenzyl)-N-methylcarboxamidoadenosine |
| AC | Adenylate Cyclase |
| ADMET | Absorption, Distribution, Metabolism, Excretion, Toxicity |
| Ado | Adenosine |
| AR | Adenosine Receptor |
| BSA | Bovine Serum Albumin |
| CCPA | 2-Chloro-N6-cyclopentyladenosine |
| CHO | Chinese Hamster Ovary |
| CPA | N6-Cyclopentyladenosine |
| DPCPX | 8-Cyclopentyl-1,3-dipropylxanthine |
| EL | Extracellular loop |
| EtOAc | Ethyl Acetate |
| DMF | Dimethylformamide |
| DMSO | Dimethylsulfoxide |
| EDTA | Ethylendiaminotetracetic Acid |
| HEPES | 4-(2-Hydroxyethyl)-1-piperazine-1-ethane sulfonic Acid |
| MOE | Molecular operating environment; |
| NECA | 5′-(N-Ethylcarboxamido)adenosine |
| rt | room temperature |
| SARs | Structure-Activity Relationships |
| THF | Tetrahydrofuran |
| TM | Transmembrane |