Table 1.
Compound | -R | MIC of (µg/mL) | |
---|---|---|---|
PAGUg1927 | PAGUg1931 | ||
GM2 | - | 1024 | 8 |
Ber3 | - | >512 | >512 |
1 | -H | 256 | 128 |
2 | o-Br | 256 | 128 |
3 | p-Br | 128 | 64 |
4 | o-F | 512 | 256 |
5 | o-Cl | 256 | 128 |
6 | p-Cl | 256 | 128 |
7 | o-CH3 | 512 | 256 |
8 | m-CH3 | 256 | 128 |
9 | p-CH3 | 256 | 128 |
10 | o-NO2 | 512 | 256 |
11 | 2,6-Cl | 128 | 64 |
Note: R, side chain of the benzyl group of 13-benzylberberine derivatives; GM, gentamicin; Ber, berberine.