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. 2020 Jan 20;20:17. doi: 10.1186/s12866-020-1706-1

Table 5.

Drug Susceptibility Profiles of patients with HIV Drug Resistance Mutations Detected

Patient No. Regimen Drug Resistance Mutation Types Susceptibility to 1 L Drugs Susceptibility to 2 L Drugs 2 L GSS Subtype
NRTIs NNRTIs PIs ABC AZT FTC 3TC TDF EFV ETR NVP RPV DRV/r ATV/r LPV/r
1 bOthers/FTC/NVP None V90I K20I S S aS S aS S S aS S S S S 3.0 02_AG
2 TDF/FTC/NVP None V90IV K20I S S aS S aS S S aS S S S S 3.0 02_AG
3 AZT/3TC/EFV None None M46 L, K20I S aS S aS S aS S S S S S S 2.75 G
4 #Others/3TC/EFV None None L10I, L23IL S aS S aS S *S S S S S S S 3.0 A1
5 AZT/3TC/NVP None E138EG None S aS S aS S S S *S L S S S 3.0 C
6 TDF/FTC/EFV None K103Q, E138AE K20I S S aS S aS aS S S L S S S 3.0 G
7 AZT/3TC/NVP None V90IV, V108IV None S aS S aS S S S aL S S S S 3.0 J
8 AZT/3TC/NVP None V108I K20I S aS S aS S S S aL S S S S 3.0 G
9 AZT/3TC/EFV None K103 N K20I S aS S aS S aH S H S S S S 3.0 G
10 AZT/3TC/EFV None V106A, F227 L K20I S aS S aS S aH S H S S S S 3.0 02_AG
11 bOthers/FTC/NVP None K103KN K20I S S aS S aS H S aH S S S S 3.0 02_AG
12 TDF/FTC/NVP None V90I, K103 N K20I S S aS S aS H S aH S S S S 3.0 02_AG
13 AZT/3TC/NVP M184 V K103 N, E138A K20I L aS H aH S H S aH L S S S 2.0 G
14 AZT/3TC/EFV D67DN, K70R, M184 V, K219E K103 N, V108I K20I L aL H aH L aH S H S S S S 1.5 02_AG
15 TDF/3TC/EFV K70E, M184 V K103 N, V108I, H221Y L10I, K20I L S H aH aL aH S H S S S S 2.0 02_AG
16 AZT/3TC/NVP M184 V A98AG, K101E, Y181C K20I L aS H aH S L L aH H S S S 2.0 02_AG

S Susceptible and Potential low-level resistance, L Low-level resistance and Intermediate-level resistance, H High-level resistance. NRTIs Nucleoside Reverse Transcriptase Inhibitors, NNRTIs Non-Nucleoside Reverse Transcriptase Inhibitors, PIs Protease Inhibitors; 1 L-First-line; 2 L = Second-line: GSS Genotype Sensitivity Score. aIndicate drugs in patient’s First-line regimen; bOthers = Backbone NRTI was switched