Skip to main content
. 2019 Dec 5;26(2):390–395. doi: 10.1002/chem.201904168

Scheme 5.

Scheme 5

Dearomatisation of C2‐ and C3‐substituted indoles: synthesis of ortho‐formyl/acyl anilide derivatives. Reaction conditions: substrate (0.25 mmol), RB (3 mol %), K3PO4 (50 mol %), DMF (0.9 mL), H2O (0.1 mL), reaction time 45 h; isolated yields. [a] Without K3PO4.