Table 3.
Effects of LND and PTX
GluCl receptor | LND | PTX | ||||||
---|---|---|---|---|---|---|---|---|
IC50 (μM) | nH | %Inhib. | n | IC50 (μM) | nH | %Inhib. | n | |
b1 | 8.0 ± 1.0 | 1.2 ± 0.1 | 65 ± 5 | 6 | 23 ± 3 | 1.1 ± 0.1 | 80 ± 9 | 6 |
c | 5.8 ± 1.3 | 1.6 ± 0.4 | 95 ± 1* | 6 | 7.1 ± 0.2* | 1.5 ± 0.1 | 97 ± 1* | 6 |
Note. Values are means ± SEM.
P < .05, significantly different from b1 GluCl receptors for the equivalent experiment.