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. 2019 Dec 30;25(1):147. doi: 10.3390/molecules25010147
FBDD fragment-based drug discovery
STD saturation transfer difference
rSTD% relative saturation transfer difference
NMR nuclear magnetic resonance
HSQC heteronuclear single quantum correlation
SAR structure activity relationship
BrmGRX Brucella melitensis glutaredoxin
hGRX1 human glutaredoxin 1
PaGRX Pseudomonas aeruginosa glutaredoxin
HTS high throughput screening
logP log of partition-coefficient
Kd dissociation constant
L.E. ligand efficiency
CSPs chemical shift perturbations
trNOE transferred nuclear overhauser effect