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. 2020 Jan 22;10:1582. doi: 10.3389/fphar.2019.01582

Table 2.

Results of PDE4 in vitro inhibition.

PDE4A
Compound (10 µM) % Inhibition
Roflumilast 100 ± 9,58
Compound 1 49,8 ± 7,66
PDE4B
Compound (10 µM) % Inhibition
Roflumilast 85,7 ± 0,68
Compound 1 100 ± 0