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. Author manuscript; available in PMC: 2020 Jan 29.
Published in final edited form as: Bioorg Med Chem Lett. 2017 Aug 12;27(18):4383–4388. doi: 10.1016/j.bmcl.2017.08.020

Table 3.

In vitro hTRPV1 antagonistic activities for α-substituted acetamide derivatives.

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WE: weakly active (17: 46%, 18: 12%, 19: 49% inhibition% at 5 μM).