Figure 1.
Synthetic route to the amide analogs 1–4, 6, 7, 9–24, 26–66. Reagents and conditions: (A) PCl3, toluene, reflux. (B) CDI, THF, reflux. (C) mw, 160 °C. For R1, R2, and R3 see Table 1.
Synthetic route to the amide analogs 1–4, 6, 7, 9–24, 26–66. Reagents and conditions: (A) PCl3, toluene, reflux. (B) CDI, THF, reflux. (C) mw, 160 °C. For R1, R2, and R3 see Table 1.