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. 2020 Feb 12;10:1648. doi: 10.3389/fphar.2019.01648

Table 2.

Comparison between the IC50 values obtained from the inversion procedure and values found in literature.

Nifedipine Lidocaine Cisapride Flecainide Verapamil
CaL Inversion 38 nM 3400 μM 775 nM 9 μM 495 nM
Literature 12 nM (Kramer et al., 2013) 11 800 nM (Kramer et al., 2013) 26 μM (Crumb et al., 2016) 202 nM (Crumb et al., 2016)
60 nM (Di Stilo et al., 1998) 27 μM (Kramer et al., 2013) 200 nM (Kramer et al., 2013)
100 nM (Mirams et al., 2011)
NaL Inversion 23 600 nM 4.3 μM 120 nM 47 μM 23 000 nM
Literature 11 μM (Crumb et al., 2016) 19 μM (Crumb et al., 2016)
Kr Inversion 40 200 nM 50 000 μM 13 nM 1.9 μM 2150 nM
Literature 440 000 nM (Kramer et al., 2013) 12 nM (Crumb et al., 2016) 0.7 μM (Crumb et al., 2016) 499 nM (Crumb et al., 2016)
275 000 nM (Zhabyeyev et al., 2013) 20 nM (Kramer et al., 2013) 1.5 μM (Kramer et al., 2013) 250 nM (Kramer et al., 2013)
6.5 nM (Mohammad et al., 1997) 143 nM (Zhang et al., 1999)