Table 3.
Pharmacokinetic profile of I-11.
| Parameter | i.v.a | Parameter | p.o.b |
|---|---|---|---|
| Cmax (ng/mL) | 7180 | Tmax (h) | 0.500 |
| t1/2 (h) | 1.20 | Cmax (ng/mL) | 654 |
| AUClast (h·ng/mL) | 2602 | t1/2 (h) | 2.50 |
| AUCINF (h·ng/mL) | 2629 | AUClast (h·ng/mL) | 1302 |
| MRTINF (h) | 0.554 | AUCINF (h·ng/mL) | 1369 |
| Vss (L/kg) | 0.213 | VZ/F (L/kg) | 12.5 |
| CL (L/h/kg) | 0.384 | CL/F (L/h/kg) | 3.83 |
| F (%) | 10.4 |
Dosed intravenously at 1 mg/kg.
Dosed orally at 5 mg/kg.