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. 2019 Sep 5;10(3):512–528. doi: 10.1016/j.apsb.2019.08.009

Table 3.

Pharmacokinetic profile of I-11.

Parameter i.v.a Parameter p.o.b
Cmax (ng/mL) 7180 Tmax (h) 0.500
t1/2 (h) 1.20 Cmax (ng/mL) 654
AUClast (h·ng/mL) 2602 t1/2 (h) 2.50
AUCINF (h·ng/mL) 2629 AUClast (h·ng/mL) 1302
MRTINF (h) 0.554 AUCINF (h·ng/mL) 1369
Vss (L/kg) 0.213 VZ/F (L/kg) 12.5
CL (L/h/kg) 0.384 CL/F (L/h/kg) 3.83
F (%) 10.4
a

Dosed intravenously at 1 mg/kg.

b

Dosed orally at 5 mg/kg.