Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Selectivity of cannabinoid antagonists. Illustrated are calculated occupancies of CB1 and CB2 cannabinoid receptors expressed as a % of total at ligand concentrations of 100 nM. Indicated are three CB1-selective antagonists, rimonabant, AM251 and LY320135 (Felder et al., 1995, 1998; Lan et al., 1999) and two CB2-selective antagonists, AM630 and SR144528 (Rinaldi-Carmona et al., 1998; Ross et al., 1999).
