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. 2020 Feb 15;12(2):618–632.

Table 1.

Functions and molecular mechanism of CUL5 in normal cells

Effectors/Targets Mechanism Function Reference
CUL5 pYCas CUL5↑/pYCas↑/FAs↑ inhibiting migration [34]
Dab-1 CUL5↑/Dab-1↑/Src↑, Fyn↓ and Reln↓ decelerating neuron migration, cortical layering [46]
Rpb1 CUL5↑/Rpb1↓ responding to DNA damage [35]
AC CUL5↑/AC↓/cAMP↓ inhibiting proliferation [36,54,55]
MAPK CUL5↑/MAPK↓ inhibiting proliferation [20]
DDA3 CUL5↑/DDA3↓/stabilize MT inhibiting proliferation [9]
β-TrCP1 CUL5↑/β-TrCP1↓ inhibiting cell growth [59]
AQP-1/2 CUL5↑/AQP-1/2↓ balancing hydrosalinity [21,22]
DEPTOR CUL5↑/DEPTOR↓ inhibiting autophagy [39]

↑: upregulation; ↓: downregulation; CUL5: cullin-5; pYCas: phosphorylated Cas; FAs: focal adhesions; Dab-1: Disabled-1; Reln: Reelin; Rpb1: RNA polymerase II’s largest subunit; MAPK: mitogen-activated protein kinase; MT: microtubule; DDA3: differential display and activation by P53, also known as PSRC1; β-TrCP: β transducin repeat-containing protein; AQP: aquaporin; DEPTOR: DEP domain-containing mTOR-interacting protein.