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. 2020 Feb 15;12(2):618–632.

Table 2.

Functions and molecular mechanism of CUL5 in cancer cells

Type Molecule Mechanism Function Reference
CUL5 Gastric cancer miR-19a, ANKRD9 miR-19a↑/ABKRD9-Elongin BC-CUL5↓ promoting proliferation, invasion and anchorage-independent growth [25,73]
Hepatocellular carcinoma (associated with HBV infection) miR-145 miR-145↓/CUL5↑ inhibiting apoptosis [31]
Hepatocellular carcinoma (not associated with HBV infection) miR-7 miR-7↓/CUL5↓ Formation of a malignant phenotype in HCC [27]
Endometrial adenocarcinoma miR-182 miR-182↑/CUL5↓ promoting proliferation [28]
Cervical cancer miR-19a/b miR-19a/b↑/CUL5↓ promoting proliferation and invasion [25]
Ovarian cancer miR-27a miR-27a↑/CUL5↓ inhibiting G2/M blockade [26]
B cell chronic lymphocytic leukemia - Chromosome region 11q22-q23↓/CUL5↓ inducing apoptosis resistance [24]
Acute promyelocytic leukemia - CUL5↑ regulating granulocyte differentiation [82]
Breast cancer - CUL5↓ promoting proliferation [29,83-85]
Angiosarcoma circ_0024169 circ_0024169 / CUL5 ratio↓ acting as a diagnostic biomarker [87]
Clear cell renal cell carcinoma - CUL5↓ increasing DNA damage, promoting mitotic disorder [88]
Small-cell lung cancer SOCS3 integrinβ1 SOCS3↓/CUL5↓/integrinβ1↑ promoting metastasis [23]
Non-small-cell lung cancer UBE2F UBE2F↑/activate CRL5/Noxa↓ inhibiting apoptosis [15]

-: no data; ↑: upregulation; ↓: downregulation; miR: microRNA; ANKRD9: ankyrin repeat domain-containing protein 9; circ: circRNA; SOCS: suppressor of cytokine signaling; UBE2F: ubiquitin conjugating enzyme E2 F.