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. 2020 Apr;72(2):466–485. doi: 10.1124/pr.119.018762

TABLE 2.

Tissue and subcellular distribution of monocarboxylate transporters

Transporter Unigene Name Tissue Distribution Subcellular Localization Expression Species References
MCT1 SLC16A1 Ubiquitous Apical and basolateral membrane Human Halestrap and Meredith, 2004; Gill et al., 2005
MCT2 SLC16A7 Liver Basolateral membrane Protein Human Garcia et al., 1994; Lin et al., 1998; Halestrap and Meredith, 2004; Wilson et al., 2005; Becker et al., 2010b
Kidney Basolateral membrane Protein Human
Apical Mouse
Skeletal muscle Protein Human
Heart Protein Human
Brain Protein Human
Spleen Protein Human
Testis Basolateral membrane Protein Human
Pancreas Protein Human
MCT3 SLC16A8 Retinal pigment epithelium Basolateral membrane Halestrap and Meredith, 2004
MCT4 SLC16A3 Kidney Basolateral membrane Protein Human Dimmer et al., 2000; Halestrap and Meredith, 2004; Settle et al., 2004; Gill et al., 2005; Wang et al., 2006b
Skeletal muscle Protein Human
Intestine Basolateral membrane Protein Human
Heart Protein Human
Lung Protein Human
MCT5 SLC16A4 Liver mRNA Rat Felmlee
Kidney mRNA Rat
MCT6 SLC16A5 Kidney mRNA Rat Felmee
Intestine Basolateral membrane Protein Human Gill et al., 2005
MCT7 SLC16A6 Kidney mRNA Rat Felmlee
MCT8 SLC16A2 Liver Sinusoidal membrane mRNA Human, Rat Bonen et al., 2006; Nishimura and Naito, 2008; Roberts et al., 2008
Kidney Basolateral membrane (proximal tubule) mRNA Human, Rat Felmlee
Adrenal gland mRNA Human
Brain (neurons, blood brain barrier) mRNA Human
Choroid plexus Apical membrane Protein Human
Mouse
Ovary mRNA Human
Thyroid gland mRNA Human
Uterus mRNA Human
Placenta mRNA Human
Heart mRNA Human
Protein Rat
Lung mRNA Rat
MCT10 SLC16A10 Liver mRNA Rat Felmlee
Kidney mRNA Rat
Intestine mRNA Rat
Lung mRNA Rat
MCT11 SLC16A11 Liver mRNA Rat Felmlee
Kidney mRNA Rat
Lung mRNA Rat
MCT12 SLC16A12 Liver mRNA Rat Felmlee
Kidney mRNA Rat
Lung mRNA Rat
MCT13 SLC16A13 Liver mRNA Rat Felmlee
Kidney mRNA Rat
Intestine mRNA Rat
Lung mRNA Rat
MCT14 SLC16A14 Peripheral blood mononuclear cells mRNA Human Banerjee et al., 2017
Kidney mRNA Rat Felmlee