Table 1.
List of the known P-gp substrates and inhibitors.
| P-gp Substrates | P-gp Inhibitors |
|---|---|
| Vincristine | Verapamil |
| Vinblastine | Cyclosporin A |
| Etoposide | Tamoxifen |
| Mitomycin C | Megestrol acetate |
| Paclitaxel | Quinine |
| Topotecan | Azodipin |
| Actinomycin D | Flupentixol |
| Doxorubicin | Valspodar |
| Daunorubicin | Dofequidar |
| Mitoxantrone | Tesmilifene |
| Epirubicin | Zosuquidar |
| Tariquidar |