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The results of in vitro plasma stability, microsomal stability, and CYP inhibition.
| M.W. | Human plasma stability (% remaining after 30 min and 2 h) | Human liver microsomal stability (% remaining after 30 min) | CYP (% of control activity @ 10 μM) | |||
|---|---|---|---|---|---|---|
| 3A4 | 2D6 | 1A2 | ||||
| TIPTP (2) | 437.44 | 97.4 and 93.8 | 4.4 | 76.6 | 98.2 | 45.7 |
