. 2019 May 6;11(3):266–271. doi: 10.1021/acsmedchemlett.9b00065

Table 2. Hinge Binder and Phenyl Linker SAR^a^,^b.

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HTRF assay protocol details are provided in the Supporting Information.

Assay results are the average of at least two replicates, and IC₅₀ determination occurred after 60 min incubation.

Assay results are N of 1.

Full length construct used in assay instead of kinase domain.

Table 2. Hinge Binder and Phenyl Linker SARa,b.