Table 4.
In vitro Biological Activity of Compounds 1 – 12.
| compound |
P. falciparum Dd2 (μM) |
A2780 (μM) |
|---|---|---|
| 1 | 0.170 ± 0.004 | 0.223 ± 0.019 |
| 2 | 0.244 ± 0.005 | 0.241 ± 0.019 |
| 3 | 18.2 ± 0.4 | NT |
| 5 | > 100 | > 10 |
| 7 | > 30 | > 10 |
| 8 | NA | > 10 |
| 9 | ~ 30 | > 10 |
| 10 | ~ 30 | > 10 |
| 11 | > 100 | > 10 |
| 12 | NA | > 10 |
| artemisinin | 0.0065 ± 0.0005 | NT |
| paclitaxel | NT | 0.013 ± 0.001 |