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. Author manuscript; available in PMC: 2021 Mar 27.
Published in final edited form as: J Nat Prod. 2019 Oct 2;83(3):569–577. doi: 10.1021/acs.jnatprod.9b00724

Table 4.

In vitro Biological Activity of Compounds 112.

compound P. falciparum
Dd2 (μM)
A2780 (μM)
1 0.170 ± 0.004 0.223 ± 0.019
2 0.244 ± 0.005 0.241 ± 0.019
3 18.2 ± 0.4 NT
5 > 100 > 10
7 > 30 > 10
8 NA > 10
9 ~ 30 > 10
10 ~ 30 > 10
11 > 100 > 10
12 NA > 10
artemisinin 0.0065 ± 0.0005 NT
paclitaxel NT 0.013 ± 0.001