Table 2.
In vitro inhibitory activities plant AHAS and their herbicidal activities.
| Compound |
A. thaliana AHAS inhibition (%) |
Rape root test (%) B. campestris |
||
|---|---|---|---|---|
| 100 μM | 10 μM | 100 mg/L | 10 mg/L | |
| 6–1 | 86.5 | 34.5 | 26.2 | 2.2 |
| 6–2 | 79.3 | 19.8 | 17.4 | 0 |
| 6–3 | 74.7 | 40.3 | 14.3 | 0 |
| 6–4 | 66.7 | 51.6 | 51.6 | 0 |
| 6–5 | 71.2 | 59.2 | 60.3 | 4.6 |
| 6–6 | 71.3 | 44.9 | 16.6 | 0 |
| 6–7 | 85.5 | 57.3 | 14.0 | 0 |
| 6–8 | 15 | 11.5 | 8.5 | 0 |
| 6–9 | 63.3 | 42.9 | 54.2 | 41.8 |
| 6–10 | 89.6 | 43.2 | 60.3 | 28.4 |
| 6–11 | 98.3 | 53.1 | 25.0 | 0 |
| 6–12 | 10 | 0 | 5 | 0 |
| 6–13 | 100 | 43.6 | 40 | 34.4 |
| 6–14 | 68.6 | 3.3 | 33.3 | 1.6 |
| 6–15 | 59.6 | 5.5 | 24.2 | 0 |
| 6–16 | 19 | 12 | 55.1 | 5.2 |
| 6–17 | 18.7 | 13.8 | 27.6 | 0 |
| 6–18 | 15.3 | 12.6 | 58.2 | 0 |
| 6–19 | 30 | 22.4 | 34.3 | 0 |
| 6–20 | 75.5 | 21.8 | 16.5 | 4.0 |
| 6–21 | 81.7 | 73.3 | 20.3 | 8 |
| 6–22 | 100 | 70.1 | 86 | 72.0 |
| 6–23 | 100 | 34 | 54.5 | 0 |
| 6–24 | 100 | 61 | 93.6 | 80.7 |
| 6–25 | 100 | 40 | 82.2 | 48.0 |
| 6–26 | 100 | 31.4 | 73.4 | 30.6 |
| 6–27 | 100 | 48.9 | 26.4 | 0 |
| 6–28 | 91.6 | 18 | 66.1 | 12.3 |
| 6–29 | 85.5 | 51.8 | 50.0 | 24.6 |
| 6–30 | 86.2 | 51.2 | 33.5 | 4.7 |
| 6–31 | 77.4 | 37.7 | 45.2 | 0 |
| 6–32 | 72.3 | 28.2 | 25.8 | 0 |
| 6–33 | 20 | 5 | 0 | 0 |
| 6–34 | 60 | 6.6 | 87.4 | 32.5 |
| 6–35 | 84.7 | 8.9 | 88.1 | 80.2 |
| Pyrithiobac | 100 | 96 | 97.0 | 90.2 |