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. 2008 Oct 11;49(51):7243–7245. doi: 10.1016/j.tetlet.2008.10.032

Table 1.

Synthesis of flavonol

Acetophenone (1)
Benzaldehyde (2)
Chalcone (3)
Flavonol (4)
R1 R2 R3 R4 R5 Yield (%) Yield (%)
a H H OMe OMe H 50 70
b H H H OMe H 60 73
c H OMe H H H 46 74
e H H OMe H H 53 69
f H H OMe OMe OMe 35 38
g H OMe H H OMe 38 45
h H OMe H OMe H 65 55
i H H H OBn H 72 71a
j H H OMe OBn H 75 80a
k OMe H OMe OMe H 30 69
l OMe H H OMe H 56 69
m OMe H OMe H H 20 59
n OMe OMe OMe H H 72 62
o OBn H H OMe H 54 76a
a

Dioxane/ethanol mixture was used as solvent.