Table 1.
Acetophenone (1) |
Benzaldehyde (2) |
Chalcone (3) |
Flavonol (4) |
||||
---|---|---|---|---|---|---|---|
R1 | R2 | R3 | R4 | R5 | Yield (%) | Yield (%) | |
a | H | H | OMe | OMe | H | 50 | 70 |
b | H | H | H | OMe | H | 60 | 73 |
c | H | OMe | H | H | H | 46 | 74 |
e | H | H | OMe | H | H | 53 | 69 |
f | H | H | OMe | OMe | OMe | 35 | 38 |
g | H | OMe | H | H | OMe | 38 | 45 |
h | H | OMe | H | OMe | H | 65 | 55 |
i | H | H | H | OBn | H | 72 | 71a |
j | H | H | OMe | OBn | H | 75 | 80a |
k | OMe | H | OMe | OMe | H | 30 | 69 |
l | OMe | H | H | OMe | H | 56 | 69 |
m | OMe | H | OMe | H | H | 20 | 59 |
n | OMe | OMe | OMe | H | H | 72 | 62 |
o | OBn | H | H | OMe | H | 54 | 76a |
Dioxane/ethanol mixture was used as solvent.