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. 2010 Feb 6;66(13):2316–2321. doi: 10.1016/j.tet.2010.02.017

Table 2.

Synthesis of 3-(indol-3-yl)-3-hydroxyindolin-2-ones 3af in TMGTf or [BMIM][BF4]–LiCl ionic liquids

Entry R1 R2 Product Yield (%)
[BMIM]BF4–LiCl TMGTf
1 H H 3a 90 92
2 Me H 3b 92 93
3 H Br 3c 88 89
4 Me Br 3d 90 87
5 H F 3e 89 90
6 Me F 3f 91 89