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. 2008 Apr 25;70:89–161. doi: 10.1016/S0065-2725(08)60930-7

SCHEME 12.

SCHEME 12

R1, R2, R3 = H, alkyl, aryl, alkylamino, alkylthio, nitro, cyano, alkylsulfonyl, etc. (a) EtOCH = C(CO2Et)2, Δ; (b) Ph2O, 260 °C.