Table 1.
SARS-CoV 3CLpro inhibitory activities (Ki) of 25a–h.
Entry no. | Inhibitors | Ki (μM) | Entry no. | Inhibitors | Ki (μM) |
---|---|---|---|---|---|
25a | ![]() |
5.90 | 25e | ![]() |
1.71 |
25b | ![]() |
23.0 | 25f | ![]() |
29.0 |
25c | ![]() |
0.46 | 25g | ![]() |
9.40 |
25d | ![]() |
1.60 | 25h | ![]() |
1.20 |
SARS-CoV 3CLpro inhibitory activities (Ki) of 25a–h.
Entry no. | Inhibitors | Ki (μM) | Entry no. | Inhibitors | Ki (μM) |
---|---|---|---|---|---|
25a | ![]() |
5.90 | 25e | ![]() |
1.71 |
25b | ![]() |
23.0 | 25f | ![]() |
29.0 |
25c | ![]() |
0.46 | 25g | ![]() |
9.40 |
25d | ![]() |
1.60 | 25h | ![]() |
1.20 |