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Anti-TRPA1screening of compound 128–139 in human and rat.
| Compound No. | hTRPA1 IC50 (μM) | rTRPA1 IC50 (μM) |
|---|---|---|
| 143 | 1.8 | 1.9 |
| 144 | 2.07 | 3.39 |
| 145 | 1.1 | 0.39 |
| 146 | >10 | 9.4 |
| 147 | 0.13 | 0.02 |
| 148 | 3.1 | 3.5 |
| 149 | 0.5 | 0.071 |
| 150 | 0.71 | 0.044 |
| 151 | >10 | 2.7 |
| 152 | >10 | 0.8 |
| 153 | 0.05 | 0.011 |
| 154 | 0.07 | 0.010 |
