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. 2012 Mar 13;52:82–97. doi: 10.1016/j.ejmech.2012.03.007

Table 4.

β-hematin inhibitory assay.

Compound % Inhibitiona Compound % Inhibitiona
10a 96 10l 66
10b 100 10m 100
10c 100 10n 79
10d 89 10o 92
10e 56 10p
10f 10q 89
10g 10r 100 (2)b
10h 53 10s 94
10i 100 CQc 18b
10j 35 Quininec 324b
10k
a

The percentage inhibition at 1 mg/ml (highest concentration tested).

b

IC50 (μM).

c

Refer to text Ref. [37].